[Substituted benzo[b]thiophenes with anti-leukotriene activity]

Ceska Slov Farm. 1999 Nov;48(6):281-6.
[Article in Czech]

Abstract

The cyclizing reaction of cinnamic acid (Ia) with thionyl chloride was optimized and a series of 3-chloro-6-subst.benzo[b]thiophene-2-carbonyl chlorides Va-Vn was prepared. Chloride Va was transformed into a series of N-aryl-3-subst. (Cl, OCH3, OH) benzo[b]thiophene-2-carboxamides VII, IX, X. The drugs were subjected to an evaluation of selected antileucotriene activities in vitro and of the anti-inflammatory effect in vivo. In agreement with the assumed mechanism, inhibition of the ear inflammation is conditioned by the antileucotriene activity, whereas inhibition of the carrageen oedema is not due to this mechanism alone.

Publication types

  • English Abstract
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Cells, Cultured
  • Edema / drug therapy
  • Leukotriene Antagonists* / chemistry
  • Leukotriene Antagonists* / pharmacology
  • Leukotriene Antagonists* / therapeutic use
  • Leukotriene B4 / biosynthesis
  • Mice
  • Neutrophils / metabolism
  • Rats
  • Thiophenes* / chemistry
  • Thiophenes* / pharmacology
  • Thiophenes* / therapeutic use

Substances

  • Leukotriene Antagonists
  • Thiophenes
  • Leukotriene B4