Abstract
[formula: see text] A mild and highly efficient cyclization of beta-hydroxy amides to oxazolines is described using DAST and Deoxo-Fluor reagents. A one-pot protocol for the synthesis of oxazoles from beta-hydroxy amides is also presented.
Publication types
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Research Support, U.S. Gov't, P.H.S.
MeSH terms
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Diethylamines / chemistry*
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Fluorine / chemistry*
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Indicators and Reagents / chemistry*
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Oxazoles / chemical synthesis*
Substances
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Diethylamines
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Indicators and Reagents
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Oxazoles
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Fluorine
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diethylaminosulfur trifluoride