Mechanisms and spread of fluoroquinolone resistance in Streptococcus pneumoniae

Res Microbiol. 2000 Jul-Aug;151(6):471-3. doi: 10.1016/s0923-2508(00)00167-4.

Abstract

The development of fluoroquinolones (FQs) with enhanced activity against Streptococcus pneumoniae is a potential advance in the treatment of pneumococcal infections, particularly those due to beta-lactam-resistant pneumococci. However, FQ-resistant clinical isolates selected by the older FQs have already been reported, with mutation(s) in both FQ targets conferring cross-resistance to newer FQs. It is likely that recombinational events between topoisomerase genes from related species of streptococci contribute to the spread of FQ resistance in S. pneumoniae. A scenario resembling that of the worldwide spread of resistance to beta lactams should be anticipated.

Publication types

  • Review

MeSH terms

  • Anti-Infective Agents / pharmacology*
  • Bacterial Proteins / drug effects
  • DNA Topoisomerase IV
  • DNA Topoisomerases, Type II / drug effects
  • DNA Topoisomerases, Type II / genetics
  • Drug Resistance, Microbial
  • Fluoroquinolones
  • Genes, Bacterial
  • Humans
  • Mutation
  • Pneumococcal Infections / epidemiology*
  • Pneumococcal Infections / microbiology*
  • Streptococcus pneumoniae / drug effects*
  • Streptococcus pneumoniae / enzymology
  • Streptococcus pneumoniae / genetics

Substances

  • Anti-Infective Agents
  • Bacterial Proteins
  • Fluoroquinolones
  • pmrA protein, Bacteria
  • DNA Topoisomerase IV
  • DNA Topoisomerases, Type II