Water-soluble 99mTc-labeled dendritic novel porphyrins tumor imaging and diagnosis

Biochem Biophys Res Commun. 2001 Feb 16;281(1):32-6. doi: 10.1006/bbrc.2001.4289.

Abstract

We have synthesized two water soluble dendritic porphyrins, termed DP1 and DP2 and have successfully radiolabeled them with 99mTc. These 99mTc-labeled porphyrins were administered to C6-glioma tumor bearing Wistar rats and scintiimaging and biodistribution studies were carried out. Tumor to muscle ratios of DP1 and DP2 were 8.0 and 9.7, respectively. These molecules may have potential for tumor imaging and diagnosis and may even prove useful as photosensitizers in photodynamic therapy applications.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Animals, Newborn
  • Brain Neoplasms / diagnosis
  • Brain Neoplasms / pathology
  • Glioma / diagnosis
  • Glioma / pathology
  • Ligands
  • Models, Chemical
  • Neoplasm Transplantation
  • Neoplasms / diagnosis*
  • Neoplasms / pathology*
  • Photosensitizing Agents / pharmacology
  • Porphyrins / chemical synthesis*
  • Rats
  • Rats, Wistar
  • Technetium*
  • Tumor Cells, Cultured

Substances

  • Ligands
  • Photosensitizing Agents
  • Porphyrins
  • Technetium