Intravenous (+)-methamphetamine causes complex dose-dependent physiologic changes in awake rats

Eur J Pharmacol. 2001 Aug 24;426(1-2):81-7. doi: 10.1016/s0014-2999(01)01202-x.

Abstract

Hemodynamic and temperature dose-response relationships were characterized in freely moving rats following i.v. (+)-methamphetamine administration to mimic the rapid onset of effects experienced by many human users. Rats received saline and (+)-methamphetamine in a repeated-measures, mixed-sequence design at 22+/-1 degrees C. Significantly greater blood pressure and heart rate elevations were observed after 1.0 and 3.0 mg/kg (+)-methamphetamine vs. 0.1 and 0.3 mg/kg. The time to peak hemodynamic values and the duration of effects were significantly greater after 3.0 mg/kg vs. the lower doses. The time to peak temperatures was significantly longer after 1.0 mg/kg vs. the lower doses. Following 3.0 mg/kg, all rats experienced temperature decreases before having elevated temperatures. The duration and magnitude of the delayed temperature elevations were significantly greater after 3.0 mg/kg vs. the lower doses. In conclusion, the (+)-methamphetamine-induced hemodynamic and temperature effects were not temporally synchronized, and the complex responses were not linearly related to dose.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Blood Pressure / drug effects
  • Body Temperature / drug effects*
  • Central Nervous System Stimulants / pharmacology*
  • Diastole
  • Dose-Response Relationship, Drug
  • Heart Rate / drug effects
  • Hemodynamics / drug effects*
  • Injections, Intravenous
  • Male
  • Methamphetamine / pharmacology*
  • Rats
  • Rats, Sprague-Dawley
  • Systole
  • Time Factors
  • Wakefulness

Substances

  • Central Nervous System Stimulants
  • Methamphetamine