[Cytosine diaminase/5-flurocytosine mediated inhibiting effect on the growth of human pancreatic carcinoma cells]

Zhongguo Yi Xue Ke Xue Yuan Xue Bao. 2000 Apr;22(2):139-43.
[Article in Chinese]

Abstract

Objective: To study the inhibition effect of E. coli cytosine diaminase (CD)/5-flurocytosine (5-FC) system on the growth of human pancreatic carcinoma cell line cells.

Methods: Recombinant retroviral vector expressing CD genes was transduced into pancreatic carcinoma cell line cells. In vitro and in vivo prodrug sensitivity assays were carried out, including: (1) detection of growth and colony forming inhibition rate of transduced cells in the presence of 5-FC; (2) observation of bystander effect by MTT method; (3) observation of the growth inhibition effect of 5-FC on transduced cell xenografts in nude mice.

Results: The growth and colony forming inhibition rate of the transduced cells in the presence of 5-FC were 80.0% and 79.0%, which were obviously higher than 4.8% and 5.0% (P < 0.01) of nontransduced cells. Mixed cells containing only 10% of transduced cells showed 50.7% reduction of proliferation (bystander effect). The growth of transduced cells xenografts could be totally regressed by 5-FC.

Conclusions: CD/5-FC system is a potential gene therapy strategy for pancreatic carcinoma.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Cell Division / drug effects
  • Cytosine Deaminase / genetics*
  • Escherichia coli / enzymology*
  • Female
  • Flucytosine / pharmacology*
  • Gene Transfer Techniques
  • Genetic Therapy
  • Genetic Vectors
  • Humans
  • Mice
  • Mice, Inbred BALB C
  • Mice, Nude
  • Neoplasm Transplantation
  • Pancreatic Neoplasms / pathology
  • Pancreatic Neoplasms / therapy*
  • Prodrugs / pharmacology*
  • Retroviridae / genetics
  • Tumor Cells, Cultured

Substances

  • Prodrugs
  • Flucytosine
  • Cytosine Deaminase