Human prostaglandin EP3 receptor isoforms show different agonist-induced internalization patterns

FEBS Lett. 2004 Aug 13;572(1-3):271-5. doi: 10.1016/j.febslet.2004.06.089.

Abstract

The human prostaglandin EP3 receptor comprises eight isoforms that differ in carboxyl-tail. We show here that the isoforms are trafficked differently. When expressed in HEK293 cells, the isoforms located to the cell surface, although a fraction of some remained in the cell. Upon prostaglandin E(2) stimulation, EP3.I internalized almost completely, EP3.II, EP3.V, EP3.VI and EP3.f internalized to a lesser extent and EP3.III and EP3.IV did not internalize. Both EP3.I and EP3.f internalized with beta-arrestin and internalization were blocked by a dominant negative form of Eps15, a clathrin-associated protein. Although EP3.II internalized, beta-arrestin did not translocate with the receptor and internalization was not blocked by mutant Eps15. EP3.V and EP3.VI internalized to discrete areas of the cell with beta-arrestin.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Cell Line
  • DNA Primers
  • Dinoprostone / pharmacology*
  • Female
  • Humans
  • Kidney
  • Mutagenesis, Site-Directed
  • Protein Isoforms / agonists
  • Protein Isoforms / genetics
  • Protein Isoforms / metabolism
  • Protein Transport
  • Receptors, Prostaglandin E / agonists
  • Receptors, Prostaglandin E / genetics
  • Receptors, Prostaglandin E / metabolism*
  • Receptors, Prostaglandin E, EP2 Subtype
  • Receptors, Prostaglandin E, EP3 Subtype
  • Recombinant Proteins / metabolism
  • Restriction Mapping
  • Transfection
  • Uterus

Substances

  • DNA Primers
  • PTGER2 protein, human
  • PTGER3 protein, human
  • Protein Isoforms
  • Receptors, Prostaglandin E
  • Receptors, Prostaglandin E, EP2 Subtype
  • Receptors, Prostaglandin E, EP3 Subtype
  • Recombinant Proteins
  • Dinoprostone