Direct demonstration of carbamoyl phosphate formation on the C-terminal domain of carbamoyl phosphate synthetase

Protein Sci. 2005 Jan;14(1):37-44. doi: 10.1110/ps.041041305. Epub 2004 Dec 2.

Abstract

Carbamoyl phosphate synthetase synchronizes the utilization of two ATP molecules at duplicated ATP-grasp folds to catalyze carbamoyl phosphate formation. To define the dedicated functional role played by each of the two ATP sites, we have carried out pulse/labeling studies using the synthetases from Aquifex aeolicus and Methanococcus jannaschii, hyperthermophilic organisms that encode the two ATP-grasp folds on separate subunits. These studies allowed us to differentially label each active site with [gamma-(32)P]ATP and determine the fate of the labeled gamma-phosphate in the synthetase reaction. Our results provide the first direct demonstration that enzyme-catalyzed transfer of phosphate from ATP to carbamate occurs on the more C-terminal of the two ATP-grasp folds. These findings rule out one mechanism proposed for carbamoyl phosphate synthetase, where one ATP acts as a molecular switch, and provide additional support for a sequential reaction mechanism where the gamma-phosphate groups of both ATP molecules are transferred to reactants. CP synthesis by subunit C in our single turnover pulse/chase assays did not require subunit N, but subunit N was required for detectable CP synthesis in the traditional continuous assay. These findings suggest that cross-talk between domain N and C is required for product release from subunit C.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Adenosine Triphosphate / chemistry
  • Bacteria / enzymology
  • Carbamoyl-Phosphate Synthase (Glutamine-Hydrolyzing) / chemistry*
  • Carbamoyl-Phosphate Synthase (Glutamine-Hydrolyzing) / isolation & purification
  • Carbamyl Phosphate / chemical synthesis*
  • Catalysis
  • Enzyme Activation
  • Methanococcus / enzymology
  • Protein Folding
  • Protein Structure, Tertiary

Substances

  • Carbamyl Phosphate
  • Adenosine Triphosphate
  • Carbamoyl-Phosphate Synthase (Glutamine-Hydrolyzing)