Clomipramine increases the incidence and duration of spike-wave discharges in freely moving WAG/Rij rats

Epilepsy Res. 2010 Jun;90(1-2):167-70. doi: 10.1016/j.eplepsyres.2010.02.011. Epub 2010 Mar 17.

Abstract

Purpose: The noradrenergic and serotonergic system may have a role in modulation of absence seizures. We investigated whether the single injection of monoamine reuptake inhibitor clomipramine has an acute effect on spike-wave discharge (SWD) activity in Wistar Albino Glaxo/Rijswijk (WAG/Rij) rats.

Methods: We injected a single dose of 20 or 50 mg/kg clomipramine intraperitoneally into WAG/Rij rats and measured the incidence and duration of SWD episodes for 4h after injection. The changes in SWDs were compared to the preceding 5-day average control level.

Results: The 20 mg/kg clomipramine significantly increased the incidence of SWDs in the first measured hour while the 50 mg/kg dose significantly increased the incidence and duration of SWDs in the whole measured 4-h period.

Conclusions: Clomipramine, by acutely elevating synaptic monoamine levels, could exacerbate absence seizures.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Analysis of Variance
  • Animals
  • Antidepressive Agents, Tricyclic / adverse effects*
  • Clomipramine / adverse effects*
  • Dose-Response Relationship, Drug
  • Electroencephalography* / methods
  • Epilepsy, Absence / chemically induced*
  • Epilepsy, Absence / genetics
  • Incidence
  • Male
  • Rats
  • Rats, Inbred Strains
  • Time Factors

Substances

  • Antidepressive Agents, Tricyclic
  • Clomipramine