NF-kappaB and STAT3 signaling in glioma: targets for future therapies

Expert Rev Neurother. 2010 Apr;10(4):575-86. doi: 10.1586/ern.10.21.

Abstract

Glioblastoma remains the most clinically challenging tumor of the CNS, as evidenced by the dismal change in overall survival over the past 50 years. However, recent advances in high-throughput screening techniques have given rise to a wealth of new information regarding the aberrant signaling pathways that drive the tumor phenotype. Two of these so-called 'oncopathways' are NF-kappaB and JAK/STAT. This review will describe the basic mechanisms of these pathways, explore the relevance of NF-kappaB and JAK/STAT signaling in glioblastoma, and look ahead to experimental compounds that will integrate our knowledge of these pathways into existing therapies.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't
  • Review

MeSH terms

  • Animals
  • Antineoplastic Agents / therapeutic use
  • Brain Neoplasms / genetics
  • Brain Neoplasms / metabolism*
  • Brain Neoplasms / therapy
  • Glioma / genetics
  • Glioma / metabolism*
  • Glioma / therapy
  • Humans
  • NF-kappa B / genetics
  • NF-kappa B / metabolism*
  • STAT3 Transcription Factor / genetics
  • STAT3 Transcription Factor / metabolism*
  • Signal Transduction / physiology*

Substances

  • Antineoplastic Agents
  • NF-kappa B
  • STAT3 Transcription Factor