Connexin43 and pannexin1 channels in osteoblasts: who is the "hemichannel"?

J Membr Biol. 2012 Jul;245(7):401-9. doi: 10.1007/s00232-012-9462-2. Epub 2012 Jul 15.

Abstract

Osteoblasts sense and respond to mechanical stimuli in a process involving influx and release of large ions and signaling molecules. Unapposed gap junction hemichannels formed of connexin43 (Cx43) have been proposed as a major route for such exchange, in particular for release of ATP and prostaglandin E₂ (PGE₂) in osteocytes. However, we have found that Cx43-null osteoblasts have unaltered, mechanically induced PGE₂ release and ATP-induced YoPro dye uptake. In contrast, PGE₂ release in response to fluid shear stress is abolished in P2X₇ receptor (P2X₇R)-null osteoblasts, and ATP-induced dye uptake is attenuated following treatment of wild-type cells with a P2X₇R or Pannexin1 (Panx1) channel blocker. These data indicate that Panx1 channels, in concert with P2X₇R, likely form a molecular complex that performs the hemichannel function in osteoblast mechanosignaling.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • Adenosine Triphosphate / metabolism
  • Animals
  • Blotting, Western
  • Cell Line
  • Cells, Cultured
  • Connexin 43 / metabolism*
  • Connexins / metabolism*
  • Dinoprostone / metabolism
  • Gap Junctions / metabolism
  • Mice
  • Nerve Tissue Proteins / metabolism*
  • Osteoblasts / metabolism*
  • Osteocytes / metabolism
  • Receptors, Purinergic P2X7 / metabolism

Substances

  • Connexin 43
  • Connexins
  • Nerve Tissue Proteins
  • Panx1 protein, mouse
  • Receptors, Purinergic P2X7
  • Adenosine Triphosphate
  • Dinoprostone