Duck hepatitis B virus: DNA polymerase and reverse transcriptase activities of replicative complexes isolated from liver and their inhibition in vitro

Virology. 1988 May;164(1):48-54. doi: 10.1016/0042-6822(88)90618-6.

Abstract

The duck hepatitis B virus (DHBV)-associated activities of reverse transcriptase and DNA polymerase and their inhibition in vitro were studied. Replicative complexes (RCs) were isolated from DHBV-infected liver by gel chromatography followed by sucrose gradient centrifugation. The RCs were detected by dot blot hybridization, using radiolabeled cloned DHBV DNA as a probe, and by the incorporation of 32P-TTP in the presence of dATP, dCTP, dGTP, and Mg2+ (endogenous DNA polymerase activity). The endogenous DNA polymerase activity associated with RCs was further studied using exogenous templates: reverse transcriptase and DNA polymerase activities were demonstrated using as substrates 32P-TTP and poly(rA) p(dT)12 or poly(dA) p(dT)12-18, respectively. Both activities were biochemically characterized. Their inhibition by various antiviral agents was studied in vitro: actinomycin D, ara-ATP, aphidicolin, suramin, chloroquin, and phosphonoformate. Among these, suramin, chloroquin, phosphonoformate, and ara-ATP were shown to be potent inhibitors of viral reverse transcriptase and DNA polymerase. Studies are now in progress to establish their antiviral activity in vivo.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • DNA-Directed DNA Polymerase / isolation & purification*
  • Ducks
  • Hepatitis B virus / enzymology*
  • Hepatitis B virus / physiology
  • Hepatitis, Viral, Animal / metabolism
  • Liver / analysis
  • Nucleic Acid Synthesis Inhibitors
  • RNA-Directed DNA Polymerase / isolation & purification*
  • Reverse Transcriptase Inhibitors
  • Viral Proteins / isolation & purification*
  • Virus Replication

Substances

  • Nucleic Acid Synthesis Inhibitors
  • Reverse Transcriptase Inhibitors
  • Viral Proteins
  • RNA-Directed DNA Polymerase
  • DNA-Directed DNA Polymerase