Impurities in Oligonucleotide Drug Substances and Drug Products

Nucleic Acid Ther. 2017 Dec;27(6):309-322. doi: 10.1089/nat.2017.0691. Epub 2017 Nov 10.

Abstract

This white paper, which is the 10th in a series intended to address issues associated with the development of therapeutic oligonucleotides, examines the subject of product-related impurities. The authors consider chemistry and safety aspects and advance arguments in favor of platform approaches to impurity identification and qualification. Reporting, identification, and qualification thresholds suitable for product-related impurities of therapeutic oligonucleotides are proposed.

Keywords: identification; impurities; oligonucleotides; qualification.

MeSH terms

  • Animals
  • Chemistry Techniques, Analytical / methods*
  • Chemistry, Pharmaceutical / methods*
  • Drug Contamination / prevention & control*
  • Drug Design
  • Drug Industry / standards
  • Female
  • Humans
  • Limit of Detection
  • Male
  • Mice
  • Models, Animal
  • Oligonucleotides / analysis*
  • Oligonucleotides / chemical synthesis
  • Oligonucleotides / therapeutic use
  • Patient Safety / standards

Substances

  • Oligonucleotides