Chronic angiotensin-converting enzyme inhibition attenuates frailty and protects against atrial fibrillation in aging mice

Heart Rhythm. 2025 Feb;22(2):452-465. doi: 10.1016/j.hrthm.2024.07.016. Epub 2024 Jul 15.

Abstract

Background: Aging is a major risk factor for atrial fibrillation (AF); however, not all individuals age at the same rate. Frailty, which is a measure of susceptibility to adverse health outcomes, can be quantified with a frailty index (FI).

Objective: This study aimed to determine the effects of angiotensin-converting enzyme (ACE) inhibition on AF and atrial remodeling in aging and frail mice.

Methods: Aging mice were treated with the ACE inhibitor enalapril for 6 months beginning at 16.5 months of age and frailty was quantified. AF susceptibility and atrial structure and function were assessed by intracardiac electrophysiology in anesthetized mice, high-resolution optical mapping in intact atrial preparations, patch clamping in isolated atrial myocytes, and histology and molecular biology in atrial tissues.

Results: Enalapril attenuated frailty in aging mice with larger effects in females. AF susceptibility was increased in aging mice but attenuated by enalapril. AF susceptibility and duration also increased as a function of FI score. P-wave duration was increased and atrial conduction velocity was reduced in aging mice and improved after enalapril treatment. Furthermore, P-wave duration and atrial conduction velocity were strongly correlated with FI score. Atrial action potential upstroke velocity (Vmax) and Na+ current (INa) were reduced whereas atrial fibrosis was increased in aging mice. Action potential Vmax, INa, and fibrosis were improved by enalapril and also correlated with FI scores.

Conclusion: ACE inhibition with enalapril attenuates frailty and reduces AF susceptibility in aging mice by preventing atrial electrical and structural remodeling.

Keywords: ACE inhibitor; Aging; Atrial fibrillation; Fibrosis; Frailty; Ion channels.

MeSH terms

  • Aging*
  • Angiotensin-Converting Enzyme Inhibitors* / administration & dosage
  • Angiotensin-Converting Enzyme Inhibitors* / pharmacology
  • Animals
  • Atrial Fibrillation* / drug therapy
  • Atrial Fibrillation* / physiopathology
  • Atrial Fibrillation* / prevention & control
  • Atrial Remodeling* / drug effects
  • Disease Models, Animal
  • Enalapril* / pharmacology
  • Female
  • Frailty* / drug therapy
  • Frailty* / physiopathology
  • Heart Atria* / drug effects
  • Heart Atria* / physiopathology
  • Male
  • Mice
  • Mice, Inbred C57BL

Substances

  • Angiotensin-Converting Enzyme Inhibitors
  • Enalapril