The Protective Role of DUSP4 in Retinal Pigment Epithelium Senescence and Degeneration

Int J Mol Sci. 2025 Apr 15;26(8):3735. doi: 10.3390/ijms26083735.

Abstract

The retinal pigment epithelium (RPE) serves as a critical guardian of subretinal homeostasis, with its dysfunction implicated in major retinal pathologies, including age-related macular degeneration (AMD) and retinitis pigmentosa. While cellular senescence has emerged as a key driver of RPE degeneration, the molecular mechanisms underlying this process remain incompletely defined. Emerging evidence implicates dual-specificity phosphatase 4 (DUSP4) in cellular stress responses through its antioxidant and anti-inflammatory capacities, yet its role in RPE pathophysiology remains unexplored. Our study reveals a compensatory increase in DUSP4 expression during AMD-associated RPE senescence. To functionally characterize this observation, we knocked down DUSP4 in the RPE of mice via subretinal injection of AAV-shDUSP4. In a sodium iodate-induced dry AMD model, mice with DUSP4 knockdown presented more severe visual impairment than control mice did. To further investigate the molecular mechanism, stable DUSP4-knockout cell lines were constructed via CRISPR/Cas9 technology. The high expression of senescence markers in the DUSP4-knockout cell lines was reversed by DUSP4 overexpression. Furthermore, DUSP4 coordinates the modulation of cell cycle, stress response, and pro-inflammatory signaling by inhibiting the p53, p38, and NF-kB pathways. These findings establish DUSP4 as a multi-functional regulator of RPE senescence. Our work not only elucidates a novel DUSP4-dependent mechanism in AMD pathogenesis but also highlights its therapeutic potential for preserving RPE function in AMD.

Keywords: age-related macular degeneration; dual-specificity phosphatase 4; retinal pigment epithelium; senescence.

MeSH terms

  • Animals
  • Cell Line
  • Cellular Senescence* / genetics
  • Disease Models, Animal
  • Dual-Specificity Phosphatases* / genetics
  • Dual-Specificity Phosphatases* / metabolism
  • Humans
  • Macular Degeneration* / genetics
  • Macular Degeneration* / metabolism
  • Macular Degeneration* / pathology
  • Mice
  • Mice, Inbred C57BL
  • Mice, Knockout
  • Mitogen-Activated Protein Kinase Phosphatases* / genetics
  • Mitogen-Activated Protein Kinase Phosphatases* / metabolism
  • NF-kappa B / metabolism
  • Protein Tyrosine Phosphatases
  • Retinal Pigment Epithelium* / metabolism
  • Retinal Pigment Epithelium* / pathology
  • Signal Transduction

Substances

  • Dual-Specificity Phosphatases
  • Mitogen-Activated Protein Kinase Phosphatases
  • Dusp4 protein, mouse
  • DUSP4 protein, human
  • NF-kappa B
  • Protein Tyrosine Phosphatases