A Prospective Pilot Clinical Study reveals a promising non-toxic anti-biofilm activity of gentamicin-EDTA-Na₂ Central Venous Catheter Lock Solution

Int J Infect Dis. 2025 Aug:157:107933. doi: 10.1016/j.ijid.2025.107933. Epub 2025 May 12.

Abstract

Objectives: The treatment of long-term intravenous catheter-related bloodstream infections (LTIVC-related BSI) often requires catheter removal or conservative treatment using intra-catheter locks, with a 50-60% success rate. We previously demonstrated the synergistic effect of a combination of gentamicin and ethylenediaminetetraacetic acid disodium salt (EDTA-Na2) against bacterial biofilms. We conducted a phase 1/2 clinical trial to assess the tolerance and efficacy of genta-EDTA-Na2 locks for the conservative treatment of LTIVC-related BSI.

Methods: Prospective study including adult patients with monomicrobial, uncomplicated LTIVC-related BSI caused by gentamicin-susceptible coagulase-negative staphylococci, Enterobacterales, or Pseudomonas aeruginosa.

Primary objective: assess the safety and efficacy at genta-EDTA-Na2 locks at day 40 (D40) by evaluating the frequency of clinical and microbiological cure 30 days after the end of treatment (D40).

Results: Eight patients were included. Complete follow-up was obtained for seven patients, six of whom met the criteria for cure. The single patient with incomplete follow-up met all criteria for cure at D23. A single microbiological failure occurred (relapse of P. aeruginosa LTIVC-related BSI). Two patients experienced at least one serious adverse event; none were attributed to the genta-EDTA-Na2 locks.

Conclusions: Genta-EDTA-Na2, used as intra-catheter locks, may be a promising anti-biofilm candidate for evaluation in a randomized controlled trial.

Keywords: Antibiotic lock therapy; Biofilm; Totally implantable venous access port; conservative treatment.

Publication types

  • Clinical Trial, Phase II
  • Clinical Trial, Phase I

MeSH terms

  • Adult
  • Aged
  • Anti-Bacterial Agents* / administration & dosage
  • Anti-Bacterial Agents* / pharmacology
  • Anti-Bacterial Agents* / therapeutic use
  • Bacteremia* / drug therapy
  • Bacteremia* / microbiology
  • Biofilms* / drug effects
  • Catheter-Related Infections* / drug therapy
  • Catheter-Related Infections* / microbiology
  • Catheter-Related Infections* / prevention & control
  • Catheterization, Central Venous / adverse effects
  • Central Venous Catheters* / microbiology
  • Edetic Acid* / administration & dosage
  • Edetic Acid* / pharmacology
  • Edetic Acid* / therapeutic use
  • Female
  • Gentamicins* / administration & dosage
  • Gentamicins* / pharmacology
  • Gentamicins* / therapeutic use
  • Humans
  • Male
  • Middle Aged
  • Pilot Projects
  • Prospective Studies
  • Pseudomonas aeruginosa / drug effects
  • Treatment Outcome

Substances

  • Edetic Acid
  • Gentamicins
  • Anti-Bacterial Agents