Efficacy and safety of switching to long-acting cabotegravir + rilpivirine versus continuing bictegravir/emtricitabine/tenofovir alafenamide in Japanese participants: 12-month results from the phase 3b randomized SOLAR trial

J Infect Chemother. 2025 Jul;31(7):102734. doi: 10.1016/j.jiac.2025.102734. Epub 2025 May 16.

Abstract

In the phase 3b SOLAR study, switching to long-acting cabotegravir + rilpivirine (CAB+RPV LA) administered every 2 months (Q2M) was non-inferior to continuing daily oral bictegravir/emtricitabine/tenofovir alafenamide (BIC/FTC/TAF). We present a post hoc analysis of Japanese participants. SOLAR is a randomized (2:1), open-label, multicenter, non-inferiority study of virologically suppressed participants switching to CAB+RPV LA Q2M (with or without oral lead-in) versus continuing BIC/FTC/TAF. The primary endpoint was HIV-1 RNA ≥50 copies/mL at Month 12 (Snapshot algorithm). Of 670 participants (modified intention-to-treat-exposed population), 20 were from Japan (LA, n = 14; BIC/FTC/TAF, n = 6). At Month 12, no participants in either Japanese group had HIV-1 RNA ≥50 copies/mL; 86 % (12/14; 2 participants withdrew) versus 100 % (6/6) had HIV-1 RNA <50 copies/mL in the LA versus BIC/FTC/TAF groups; none had confirmed virologic failure. Withdrawals were due to a non-drug-related adverse event (AE; acute hepatitis B) and a physician decision. Excluding injection site reactions, drug-related AE rates were higher in the LA group (36 % vs 17 %; all grade 1 or 2). No drug-related serious AEs were reported. Injection site reactions were common (100 % [13/13] of LA participants); all were grade 1 or 2; none led to withdrawal; median duration was 4 days. Mean treatment satisfaction scores improved from baseline to Month 12 in the LA versus BIC/FTC/TAF Japanese groups (+6.25 vs + 0.33 on a 66-point scale). Though limited, these data suggest switching to CAB+RPV LA from BIC/FTC/TAF was well tolerated in Japanese participants, with comparable efficacy and improved treatment satisfaction. ClinicalTrials.gov; NCT04542070 (https://www.clinicaltrials.gov/study/NCT04542070).

Keywords: Cabotegravir; HIV-1; Japan; Long-acting; Rilpivirine.

Publication types

  • Randomized Controlled Trial
  • Clinical Trial, Phase III
  • Multicenter Study

MeSH terms

  • Adult
  • Alanine
  • Amides
  • Anti-HIV Agents* / administration & dosage
  • Anti-HIV Agents* / adverse effects
  • Anti-HIV Agents* / therapeutic use
  • Diketopiperazines
  • Drug Combinations
  • Drug Substitution
  • East Asian People
  • Emtricitabine / administration & dosage
  • Emtricitabine / therapeutic use
  • Female
  • HIV Infections* / drug therapy
  • HIV Infections* / virology
  • HIV-1 / drug effects
  • HIV-1 / isolation & purification
  • Heterocyclic Compounds, 3-Ring
  • Heterocyclic Compounds, 4 or More Rings / administration & dosage
  • Heterocyclic Compounds, 4 or More Rings / therapeutic use
  • Humans
  • Japan
  • Male
  • Middle Aged
  • Piperazines
  • Pyridones* / administration & dosage
  • Pyridones* / adverse effects
  • Pyridones* / therapeutic use
  • RNA, Viral / blood
  • Rilpivirine* / administration & dosage
  • Rilpivirine* / adverse effects
  • Rilpivirine* / therapeutic use
  • Tenofovir / administration & dosage
  • Tenofovir / analogs & derivatives
  • Tenofovir / analogs & derivatives
  • Tenofovir / therapeutic use
  • Treatment Outcome
  • Viral Load / drug effects

Substances

  • Alanine
  • Anti-HIV Agents
  • bictegravir
  • cabotegravir
  • Drug Combinations
  • Emtricitabine
  • Heterocyclic Compounds, 4 or More Rings
  • Pyridones
  • Rilpivirine
  • RNA, Viral
  • Tenofovir
  • tenofovir alafenamide
  • Diketopiperazines
  • Piperazines
  • Heterocyclic Compounds, 3-Ring
  • Amides

Supplementary concepts

  • Japanese people

Associated data

  • ClinicalTrials.gov/NCT04542070