Effectiveness of perampanel as only concomitant antiseizure medication for highly active epilepsy: insight from a real-world, multicenter retrospective study

J Neurol. 2025 Jun 7;272(7):449. doi: 10.1007/s00415-025-13184-z.

Abstract

Introduction: Managing patients with highly frequent seizures poses significant challenges for clinicians due to their high resistance to therapy. This study aims to evaluate the 12-month efficacy, safety, and tolerability of PER as the sole add-on therapy for patients with highly active epilepsy in a real-world setting.

Methods: Data from the previous Italian retrospective, observational, multicenter "PERampanel as Only Concomitant Antiseizure Medication" (PEROC) study were analyzed, categorizing patients by baseline seizure frequency into three groups: < 5, 5-20, and > 20 seizures/month. Retention, responder (≥ 50% seizure reduction) rates, seizure-free rates and adverse events (AEs) were analyzed. Sub-analyses examined early (≤ 1 previous ASM) vs. late (> 2 previous ASMs) add-on groups.

Results: The sample included 485 patients with focal and generalized epilepsy: 354 with < 5 seizures/month, 79 with 5-20, and 52 with > 20 seizures/month. Retention rates at 12 months were 75.1%, 68%, and 58.1.7%, respectively. Perampanel significantly reduced seizure frequency in all groups, with responder rates of 71.2%, 61.8%, and 63.2% at the 12-month follow-up. Patients with more frequent seizures (> 20 and 5-20 seizures/month) had lower seizure-free rates (15.8% and 23.5%) compared to those with < 5 seizures/month (49.5%, p = 0.001). AEs, mainly dizziness and irritability occurred in 30% of patients, without significant differences between groups (p = 0.092).

Conclusions: PER, as the sole adjunctive therapy, demonstrated good effectiveness and tolerability in a real-world setting, even for patients with highly active epilepsy. These findings suggest PER as a valuable early treatment option to improve seizure control and quality of life in this challenging population.

Keywords: Anti-seizure medication; Drug-refractory epilepsy; Early add-on; Real-world evidence; Seizure freedom; Very active epilepsy.

Publication types

  • Multicenter Study
  • Observational Study

MeSH terms

  • Adolescent
  • Adult
  • Aged
  • Anticonvulsants* / administration & dosage
  • Anticonvulsants* / adverse effects
  • Anticonvulsants* / therapeutic use
  • Drug Therapy, Combination
  • Epilepsies, Partial* / drug therapy
  • Epilepsy* / drug therapy
  • Epilepsy, Generalized* / drug therapy
  • Female
  • Humans
  • Male
  • Middle Aged
  • Nitriles
  • Pyridones* / administration & dosage
  • Pyridones* / adverse effects
  • Pyridones* / therapeutic use
  • Retrospective Studies
  • Seizures / drug therapy
  • Treatment Outcome
  • Young Adult

Substances

  • Anticonvulsants
  • perampanel
  • Pyridones
  • Nitriles