The Lemon Flavonoid Eriomin® Suppresses Pituitary-Adrenal Axis Activity in Aged Rats

Int J Mol Sci. 2025 Jun 17;26(12):5818. doi: 10.3390/ijms26125818.

Abstract

The lemon flavonoid extract Eriomin® (LE), which is rich in eriocitrin, has demonstrated antioxidant and anti-inflammatory properties in both animal and human studies. Given the established interplay among aging, oxidative stress, and inflammation, this study investigated the influences of LE on the pituitary-adrenal (PA) axis in aged rats and its potential to mitigate age-related physiological changes in this system. The effects of LE (40 mg/kg/day suspended in sunflower oil) on the morphofunctional properties of the PA axis were studied in 24-month-old male Wistar rats following four weeks of oral treatment. Control groups included vehicle-treated (sunflower oil; CON) and untreated intact controls (ICON). Stereological and imaging analyses revealed no significant changes in pituitary ACTH cells; however, Pomc gene expression was significantly downregulated in the LE group compared to both controls (p ≤ 0.05). LE treatment resulted in a significant reduction in adrenal gland weight (p ≤ 0.05), adrenal gland volume (p ≤ 0.01), zona fasciculata (ZF) volume (p ≤ 0.01) and ZF cell volume (p ≤ 0.05). These changes were accompanied by a significant decrease in serum corticosterone levels (p ≤ 0.05). In conclusion, LE downregulated PA axis activity in aged rats. Considering the association between age-related increases in PA activity and adverse health outcomes, citrus flavonoid extracts such as LE may hold promise as anti-aging supplements aimed at mitigating age-related stress dysregulation.

Keywords: adrenal gland; aged rat; healthy ageing; lemon flavonoid extract Eriomin®; pituitary gland.

MeSH terms

  • Adrenal Glands / drug effects
  • Adrenal Glands / metabolism
  • Adrenocorticotropic Hormone / metabolism
  • Aging* / drug effects
  • Animals
  • Citrus* / chemistry
  • Corticosterone / blood
  • Flavonoids* / pharmacology
  • Male
  • Pituitary-Adrenal System* / drug effects
  • Pituitary-Adrenal System* / metabolism
  • Plant Extracts* / chemistry
  • Plant Extracts* / pharmacology
  • Pro-Opiomelanocortin / genetics
  • Pro-Opiomelanocortin / metabolism
  • Rats
  • Rats, Wistar

Substances

  • Flavonoids
  • Plant Extracts
  • Corticosterone
  • Adrenocorticotropic Hormone
  • Pro-Opiomelanocortin