Inhibition of Axl attenuates acute kidney injury by alleviating inflammation via SOCS3 downregulation in tubular epithelial cells

BMC Nephrol. 2025 Jul 1;26(1):325. doi: 10.1186/s12882-025-04222-z.

Abstract

Background: In acute kidney injury (AKI), inflammatory crosstalk between tubular epithelial cells (TECs) and immune cells drives disease progression. Although the Axl-SOCS3 axis in myeloid cells typically suppresses inflammation, TEC-specific SOCS3 deletion paradoxically protects against AKI, suggesting a cell type-specific pro-inflammatory role.

Methods: We induced AKI via bilateral ischemia/reperfusion (IRI) in mice. The Axl-specific pharmacological inhibitor R428 was administered via subcutaneous injection immediately post-IRI, with plasma and kidney samples collected 24 h later. To assess the effects of SOCS3 in TECs, small interfering RNA was used to silence SOCS3 in cisplatin injured HK2 cells. Axl/SOCS3 expression levels were assessed in human AKI biopsies.

Results: In AKI patients and IRI mice, Axl was upregulated in interstitial immune cells, while SOCS3 increased in TECs. Axl inhibition by R428 attenuated renal injury, reducing inflammatory infiltration, NF-κB p65 phosphorylation, and TEC SOCS3 expression. Notably, SOCS3 knockdown in TECs suppressed NF-κB activation and IL-1β/IL-6 production, implicating Axl-SOCS3 as a pro-inflammatory amplifier in AKI.

Conclusion: The Axl-SOCS3 axis exacerbates AKI by reinforcing NF-κB-driven inflammation in TECs, creating a vicious cycle between immune cells and TECs. Targeting this cross-cellular pro-inflammatory pathway offers a promising therapeutic strategy for AKI.

Keywords: Acute kidney injury; Axl; Inflammation; Suppressor of cytokine signaling 3; Tubular epithelial cells.

MeSH terms

  • Acute Kidney Injury* / drug therapy
  • Acute Kidney Injury* / metabolism
  • Acute Kidney Injury* / pathology
  • Animals
  • Axl Receptor Tyrosine Kinase
  • Benzocycloheptenes* / pharmacology
  • Benzocycloheptenes* / therapeutic use
  • Down-Regulation / drug effects
  • Epithelial Cells* / drug effects
  • Epithelial Cells* / metabolism
  • Humans
  • Inflammation / metabolism
  • Kidney Tubules* / cytology
  • Kidney Tubules* / drug effects
  • Kidney Tubules* / metabolism
  • Kidney Tubules* / pathology
  • Male
  • Mice
  • Mice, Inbred C57BL
  • Proto-Oncogene Proteins* / antagonists & inhibitors
  • Proto-Oncogene Proteins* / metabolism
  • Receptor Protein-Tyrosine Kinases* / antagonists & inhibitors
  • Receptor Protein-Tyrosine Kinases* / metabolism
  • Reperfusion Injury / metabolism
  • Suppressor of Cytokine Signaling 3 Protein* / genetics
  • Suppressor of Cytokine Signaling 3 Protein* / metabolism
  • Triazoles

Substances

  • Suppressor of Cytokine Signaling 3 Protein
  • Receptor Protein-Tyrosine Kinases
  • Axl Receptor Tyrosine Kinase
  • Proto-Oncogene Proteins
  • Socs3 protein, mouse
  • SOCS3 protein, human
  • AXL receptor tyrosine kinase, mouse
  • Benzocycloheptenes
  • bemcentinib
  • Triazoles