Discovery and Characterization of a First-in-Class LIV1-TLR7/8 Immunomodulatory Conjugate with Robust Myeloid Activation and Antitumor Activity.
Yamazoe S, Poudel Y, Sega E, Mukhopadhyay A, Ramakrishnan R, Ukairo O, Liu S, Akter R, Sadanala K, Que K, Cheng Q, Kotapati S, Deshpande M, Cox M, Chourey S, Gupta A, Kempson J, Pabbisetty K, Kaspady M, Bhattasali D, Yip S, Wu DR, Pookot D, Li Y, Kozhich A, Drexler D, Carl S, Deyanova E, Smith M, Chan H, West S, Diong SJ, Chang A, Florin L, Mathur A, Strop P, Zapf CW, Law D, Wilson N, Broz M, Chekler EP.
Yamazoe S, et al. Among authors: deshpande m.
J Med Chem. 2025 Jun 12;68(11):11322-11339. doi: 10.1021/acs.jmedchem.5c00264. Epub 2025 May 24.
J Med Chem. 2025.
PMID: 40411528
Free PMC article.