A cereblon-based glue degrader of NEK7 regulates NLRP3 inflammasome in a context-dependent manner.
Sylvain A, Stoehr N, Ma F, Cernijenko A, Schröder M, Khoshouei M, Vogelsanger M, Schoenboerner M, Burke A, Rao P, Solomon JM, Paulk J, Xu L, Dawson J, Begue D, Lefeuvre P, Ahrne E, Hofmann A, Dickson CJ, Arabin P, Zimmerlin A, Kiffe M, Froehlicher M, Boersig T, Elhajouji A, Brichet M, Menon S, Liu S, Mueller M, Wartchow CA, Lin J, Gloria YC, Dickhöfer S, Weber ANR, Welzel T, Kuemmerle-Deschner J, Farady CJ, Pulz R, Bornancin F, Buckley DL, Bassi ZI.
Sylvain A, et al. Among authors: ma f.
Cell Chem Biol. 2025 Jul 7:S2451-9456(25)00200-4. doi: 10.1016/j.chembiol.2025.06.005. Online ahead of print.
Cell Chem Biol. 2025.
PMID: 40639372